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Search Results for " dopa decarboxylase "
Targets Recommended: Dopamine Receptor

7

抑制剂 & 化合物

2

天然产物

2

重组蛋白

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Cat. No. Product Name Target Signaling Pathways
T1517 Benserazide hydrochloride

Benserazide HCl,盐酸苄丝肼,Serazide,Ro 4-4602

Dopamine Receptor GPCR/G Protein; Neuroscience
Benserazide hydrochloride (Ro 4-4602) 是一种芳香族 L-氨基酸脱羧酶(AADC)的抑制剂,常用于帕金森病。
T2148 Carbidopa monohydrate

Carbidopa Hydrate,S(-)-Carbidopa,卡比多巴水合物

Decarboxylase; Aryl Hydrocarbon Receptor Immunology/Inflammation; Metabolism; Others
Carbidopa monohydrate (S(-)-Carbidopa) 是一种外周型脱羧酶抑制剂,可用于帕金森病的研究。它是一种选择性芳香烃受体 (AhR) 调节剂。它抑制胰腺癌细胞和肿瘤生长。
T5954 Methyldopa hydrate

L-甲基多巴,Alpha-Methyldopa Sesquihydrate,L-(-)-α-Methyldopa hydrate,MK-351 hydrate,Methyldopa Sesquihydrate

Dopamine Receptor; Adrenergic Receptor GPCR/G Protein; Neuroscience
Methyldopa hydrate (MK-351 hydrate) 是一种前药,在中枢神经系统中被代谢成 α-Methylepinephrine。它是一种 α-肾上腺素能激动剂,对α2-adrenergic receptors 有选择性。
T15701 Methyldopa hydrochloride

L-(-)-α-Methyldopa hydrochloride,MK-351 hydrochloride

Others Others
L-(-)-α-Methyldopa hydrochloride is an alpha-adrenergic agonist psychoactive drug. It is used as a sympatholytic or antihypertensive. Methyldopa has a dual mechanism of action. It is a competitive inhibitor of the enzyme DOPA decarboxylase, which converts
T20396 Levadopa Related Compound A

6-Hydroxydopa, L-,L-Hydroxydopa

Levadopa Related Compound A is the 6-hydroxy derivative of the amino acid L-DOPA with neurotoxic properties. Exogenously administered 6-Hydroxy-L-DOPA is biotransformed by an amino acid decarboxylase to the highly potent and catecholamine-selective neurot
T1517L Benserazide

Ro-44602,Ro44602,Ro 44602,Serazide

Benserazide is an inhibitor of dopa decarboxylase. It is often given with levodopa in the treatment of Parkinson's to prevent the conversion of levodopa to dopamine in the periphery, thereby increasing the amount that reaches the central nervous system an
T36207 Methylspinazarin

Methylspinazarin is a naphthoquinone bacterial metabolite that has been found in Streptomyces and is an inhibitor of catechol O-methyltransferase (COMT; IC50 = 0.8 μg/ml).1 It is selective for COMT over tyrosine hydroxylase, DOPA decarboxylase, and dopamine-β-hydroxylase at 100 μg/ml. Methylspinazarin decreases blood pressure in spontaneously hypertensive rats when administered at a dose of 50 mg/kg. |1. Chimura, H., Sawa, T., Takita, T., et al. Methylspinazarin and dihydromethylspinazarin, gate...

化合物

Benserazide hydrochloride
Cat.No: T1517
Synonym: Benserazide HCl,盐酸苄丝肼,Serazide,Ro 4-4602
Target: Dopamine Receptor
Carbidopa monohydrate
Cat.No: T2148
Synonym: Carbidopa Hydrate,S(-)-Carbidopa,卡比多巴水合物
Target: Decarboxylase, Aryl Hydrocarbon Receptor
Methyldopa hydrate
Cat.No: T5954
Synonym: L-甲基多巴,Alpha-Methyldopa Sesquihydrate,L-(-)-α-Methyldopa hydrate,MK-351 hydrate,Methyldopa Sesquihydrate
Target: Dopamine Receptor, Adrenergic Receptor
Methyldopa hydrochloride
Cat.No: T15701
Synonym: L-(-)-α-Methyldopa hydrochloride,MK-351 hydrochloride
Target: Others
Levadopa Related Compound A
Cat.No: T20396
Synonym: 6-Hydroxydopa, L-,L-Hydroxydopa
Target:
Benserazide
Cat.No: T1517L
Synonym: Ro-44602,Ro44602,Ro 44602,Serazide
Target:
Methylspinazarin
Cat.No: T36207
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
T0848 L-DOPA

左旋多巴,Levodopa,3,4-Dihydroxyphenylalanine

Dopamine Receptor; Endogenous Metabolite GPCR/G Protein; Metabolism; Neuroscience
L-DOPA (Levodopa) 是的神经递质多巴胺的代谢前体,具有口服活性。Levodopa 能够透过血脑屏障,并在大脑中转化为多巴胺。Levodopa 具有抗痛觉过敏作用。Levodopa 还具有帕金森氏病的研究潜力。
TN3607 Catalpalactone

cAMP GPCR/G Protein
Catalpalactone exhibits high antitermitic, and cytotoxic activities, it exhibits potent inhibitory effects on lipopolysaccharide-induced NO synthesis in RAW 264.7 cells , with IC50 values of 9.80 microM. Catalpalactone can inhibit dopamine biosynthesis by

天然产物

L-DOPA
Cat.No: T0848
Synonym: 左旋多巴,Levodopa,3,4-Dihydroxyphenylalanine
Target: Dopamine Receptor, Endogenous Metabolite
Catalpalactone
Cat.No: TN3607
Synonym:
Target: cAMP
Cat. No. Product Name Species Expression System
TMPY-02472 DOPA Decarboxylase/DDC Protein, Mouse, Recombinant (His)

Aadc,dopa decarboxylase (aromatic L-amino ...

Mouse Baculovirus Insect Cells
DOPA Decarboxylase/DDC Protein, Mouse, Recombinant (His) is expressed in Baculovirus insect cells with His tag. The predicted molecular weight is 55.2 kDa and the accession number is O88533.
TMPY-01060 DOPA Decarboxylase/DDC Protein, Human, Recombinant (His)

dopa decarboxylase (aromatic L-amino acid ...

Human Baculovirus Insect Cells
DOPA Decarboxylase/DDC Protein, Human, Recombinant (His) is expressed in Baculovirus insect cells with His tag. The predicted molecular weight is 55 kDa and the accession number is Q53Y41.

重组蛋白

DOPA Decarboxylase/DDC Protein, Mouse, Recombinant (His)
Cat.No: TMPY-02472
Species: Mouse
Expression System: Baculovirus Insect Cells
DOPA Decarboxylase/DDC Protein, Human, Recombinant (His)
Cat.No: TMPY-01060
Species: Human
Expression System: Baculovirus Insect Cells
TargetMol Loading
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